1 Tmax
Exposure / Absorption
20-30 minutes
1,200-1,800 seconds
TGA Product Information 5.2 pharmacokinetic properties manual extraction plasma human intramuscular 2 Tmax
Exposure / Absorption
0.25-0.75 h
900-2,700 seconds
Canadian Product Monograph 10.3 pharmacokinetics manual extraction plasma human intramuscular 3 Tmax
Exposure / Absorption
Canadian Product Monograph Table 2 pharmacokinetics manual extraction serum human intramuscular 50 mg intramuscular dose 4 Tmax
Exposure / Absorption
0.5-2 hours
1,800-7,200 seconds
Canadian Product Monograph detailed pharmacology manual extraction serum human intramuscular 5 Tmax
Exposure / Absorption
UK eMC SmPC section 5.2 pharmacokinetics manual extraction serum human subcutaneous 6 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 140 mg dose infused over 30 min 7 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 220 mg dose infused over 30 min 8 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 350 mg dose infused over 30 min 9 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 500 mg dose infused over 30 min 10 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 630 mg dose infused over 30 min 11 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 840 mg dose infused over 30 min 12 Tmax
Exposure / Absorption
FDA Clinical Pharmacology Review Table 6 manual extraction plasma human intravenous single 1120 mg dose infused over 30 min 13 Tmax
Exposure / Absorption
14 Tmax
Exposure / Absorption
15 Tmax
Exposure / Absorption
16 Tmax
Exposure / Absorption
17 Tmax
Exposure / Absorption
Peak serum levels after intravenous (i.v.) administration are achieved within 10 min. They appeared higher but declined more rapidly than those achieved after i.m. administration
Show more 18 Tmax
Exposure / Absorption
Tmax in Gottingen mini pig at 2 nmol/kg, sc porcine sc 19 Tmax
Exposure / Absorption
Tmax in cannulated Sprague-Dawley rat at 10 nmol, sc by EIA rat sc 20 Tmax
Exposure / Absorption
Tmax in Sprague-Dawley rat at 15 nmol/kg, sc by LC-MS/MS analysis rat sc